SCHEMBL9079496

SCHEMBL9079496

CS(=O)(=O)Nc1ccc(C(=O)CN2CCC(C(O)C(=O)c3ccc(F)c(F)c3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 1/20 0.43
KCNH2 Q12809 4/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
ADRA2C P18825 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
CHRM1 P11229 1/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
CYP2D6 P10635 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9077465 0.86 CYP2D6 (0.45) GRIN2BALDH1A1MAPTKCNH2MEN1
SCHEMBL9077025 0.84 KCNH2 (0.50) GRIN2BALDH1A1MAPTKCNH2MEN1
Hydrochloric Acid SCHEMBL9078685 0.83 KCNH2 (0.51) GRIN2BALDH1A1MAPTKCNH2MEN1
SCHEMBL9079349 0.79 CYP2D6 (0.58) GRIN2BALDH1A1MAPTKCNH2HTR2A
SCHEMBL9077057 0.77 CYP2D6 (0.53) MAPTKCNH2MEN1KMT2AHTR2A
SCHEMBL9076918 0.77 MEN1 (0.47) GRIN2BALDH1A1MEN1KMT2A
SCHEMBL9444257 0.74 KCNH2 (0.60) GRIN2BALDH1A1MAPTKCNH2MEN1
SCHEMBL9077056 0.74 KCNH2 (0.53) ALDH1A1MAPTKCNH2MEN1KMT2A
SCHEMBL8958724 0.74 SMN1; SMN2 (0.63) ALDH1A1KCNH2MEN1KMT2AHTR2A
SCHEMBL10646175 0.73 ALDH1A1 (0.56) GRIN2BALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532629-B1 1-PIPERIDINYL ALKANOYLARYLSULFONAMIDE DERIVATIVES MERRELL PHARMA INC (US) 1996-11-06 EP claimed