SCHEMBL9080100

SCHEMBL9080100

COc1ccc2c(c1)cc(C(=O)O)c1c(C(=O)OC(=O)c3cccc4c3c(C(=O)O)cc3cc(OC)ccc34)cccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.46
KDM4E B2RXH2 11/20 0.44
ALDH1A1 P00352 7/20 0.44
HPGD P15428 6/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
ATM Q13315 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 4/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA3 P07451 2/20 0.44
CA5A P35218 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9279459 0.92 CDC25B (0.50) CDC25BKDM4EALDH1A1HPGDNPC1
SCHEMBL9080297 0.85 MTNR1A (0.47) CDC25BKDM4EALDH1A1HPGDMAPT
SCHEMBL9079015 0.83 KDM4E (0.51) CDC25BKDM4EALDH1A1HPGDMAPT
SCHEMBL9041814 0.82 NR4A1 (0.51) CDC25BKDM4EALDH1A1HPGDMAPT
SCHEMBL9080057 0.76 ALDH1A1 (0.41) CDC25BKDM4EALDH1A1HPGDNPC1
SCHEMBL11271721 0.76 KDM4E (0.57) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL31613816 0.76 CDC25B (0.64) CDC25BKDM4EALDH1A1HPGDNPC1
SCHEMBL2510203 0.76 CDC25B (0.64) CDC25BKDM4EALDH1A1HPGDNPC1
SCHEMBL9041045 0.75 CLK1 (0.42) CDC25BKDM4EALDH1A1LMNAMAPT
SCHEMBL9077953 0.74 CNR2 (0.40) CDC25BKDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed