SCHEMBL9080180

SCHEMBL9080180

c1ccc(Oc2ccc(CNCC34CC5CC(CC(C5)C3)C4)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.54
P2RX7 Q99572 6/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
EPHX2 P34913 4/20 0.46
LTA4H P09960 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 1/20 0.43
KDM1A O60341 2/20 0.43
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067533 0.86 P2RX7 (0.67) HDAC6P2RX7MEN1KMT2AHDAC3
SCHEMBL15008930 0.79 CNR2 (0.54) HDAC6MEN1KMT2AEPHX2LTA4H
SCHEMBL18088397 0.77 HDAC6 (0.61) HDAC6P2RX7MEN1KMT2AHDAC3
SCHEMBL1160892 0.77 P2RX7 (0.55) HDAC6P2RX7MEN1KMT2AHDAC3
SCHEMBL8497858 0.76 KDM4E (0.67) MEN1KMT2AEPHX2LTA4HKDM4E
SCHEMBL7756966 0.74 KDM4E (0.70) MEN1KMT2AEPHX2LTA4HKDM4E
SCHEMBL18085885 0.74 HDAC6 (0.57) HDAC6P2RX7MEN1KMT2AHDAC3
Hydrochloric Acid SCHEMBL9079843 0.72 KDM4E (0.68) MEN1KMT2AEPHX2LTA4HKDM4E
SCHEMBL18423583 0.72 HDAC6 (0.70) HDAC6P2RX7MEN1KMT2AHDAC3
SCHEMBL10131890 0.72 P2RX7 (0.50) HDAC6P2RX7MEN1KMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996034851-A1 BENZENE, PYRIDINE, NAPHTALENE OR BENZOPHENONE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHETASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LABORATORIES (US) 1996-11-07 WO disclosed