SCHEMBL9080267

SCHEMBL9080267

O=c1[nH]c2ccc(C(F)(F)F)cc2n(Cc2ccccc2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
PGR P06401 1/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
DDR1 Q08345 4/20 0.44
HDAC11 Q96DB2 1/20 0.44
RGS4 P49798 1/20 0.44
RGS8 P57771 1/20 0.44
MDH2 P40926 1/20 0.43
GRIK1 P39086 1/20 0.43
GRIA1 P42261 1/20 0.43
GRIA2 P42262 1/20 0.43
GRIA3 P42263 1/20 0.43
GRIA4 P48058 1/20 0.43
GRIK2 Q13002 1/20 0.43
GRIK3 Q13003 1/20 0.43
GRIK4 Q16099 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30530478 0.79 APOBEC3G (0.61) CFTRKDM4EALDH1A1GRIA1GRIA2
SCHEMBL7329647 0.79 APOBEC3G (0.61) CFTRKDM4EALDH1A1GRIA1GRIA2
SCHEMBL24335163 0.77 ALDH1A1 (0.48) HDAC1HDAC8HDAC6KDM4EALDH1A1
SCHEMBL29580281 0.77 ALDH1A1 (0.48) HDAC1HDAC8HDAC6KDM4EALDH1A1
SCHEMBL29482656 0.77 KMT2A (0.48) KDM4EALDH1A1BRD4HPGDTSHR
SCHEMBL28702303 0.77 KMT2A (0.48) KDM4EALDH1A1BRD4HPGDTSHR
SCHEMBL10508287 0.75 PARG (0.53) HDAC1HDAC8HDAC6PGRKDM4E
SCHEMBL9080167 0.74 CA12 (0.52) HDAC1HDAC8HDAC6PGRKDM4E
SCHEMBL28691251 0.73 CFTR (0.52) CFTRKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL30581508 0.73 CFTR (0.52) CFTRKDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559106-A Heterocyclic compounds, their use and preparation NOVO NORDISK A/S (DK) 1996-09-24 US disclosed
EP-0691969-A1 [1,2,4] TRIAZOLO [4,3-a] QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1996-01-17 EP disclosed
WO-1994021639-A1 [1,2,4] TRIAZOLO [4,3-a] QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-09-29 WO disclosed