SCHEMBL9080434

SCHEMBL9080434

CC(C)(C)c1ccc2c(C(O[SiH3])(c3ccccc3)c3ccccc3)c(CBr)ccc2c1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.32
KIF11 P52732 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9508650 0.88 KIF11 (0.34) NR1I2KIF11CYP2D6
SCHEMBL15066839 0.67 PTPN1 (0.41) KIF11CYP2D6
SCHEMBL8954235 0.66 ALDH1A1 (0.33) KIF11CYP2D6
SCHEMBL6044524 0.64 MAOB (0.46)
SCHEMBL10409091 0.64 ALDH1A1 (0.54) NR1I2KIF11CYP2D6
SCHEMBL31012297 0.63 CYP2C19 (0.47) CYP2D6
SCHEMBL8762233 0.63 CYP2C19 (0.47) CYP2D6
SCHEMBL15067703 0.62 PTPN1 (0.44)
SCHEMBL3482515 0.62 KIF11 (0.43) KIF11
SCHEMBL8464287 0.62 CYP1A2 (0.60) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574039-A ANTITUMOR, FUNGICIDES AGOURON PHARMACEUTICALS, INC. (US) 1996-11-12 US disclosed
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed