SCHEMBL9084007

SCHEMBL9084007

COC(=O)c1ccc(OCCCN2CCC(C(=O)c3nc4ccccc4s3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 5/20 0.53
MAPT P10636 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
HRH3 Q9Y5N1 3/20 0.48
HTR1A P08908 2/20 0.48
DRD2 P14416 2/20 0.48
HTR2A P28223 2/20 0.48
SLC6A4 P31645 2/20 0.48
HTR7 P34969 2/20 0.48
MAOB P27338 1/20 0.48
HRH1 P35367 2/20 0.47
SLC6A2 P23975 1/20 0.47
HTR2C P28335 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GLO1 Q04760 1/20 0.46
MEN1 O00255 1/20 0.46
TSHR P16473 1/20 0.46
CRHBP P24387 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846152 0.90 LTA4H (0.55) LTA4HHRH3HTR1ADRD2HTR2A
SCHEMBL9398887 0.90 HRH2 (0.47) MAPTNPC1RAB9AHRH3DRD2
SCHEMBL7839234 0.86 LTA4H (0.54) LTA4HHRH3HTR1ADRD2HTR2A
SCHEMBL7839579 0.81 HRH3 (0.48) MAPTHRH3DRD2MAOBHRH1
SCHEMBL7840871 0.80 HRH3 (0.48) LTA4HHRH3MAOBHRH1HRH2
SCHEMBL7836502 0.79 HRH3 (0.47) HRH3MAOBHRH1KMT2AHRH2
SCHEMBL7828710 0.79 LTA4H (0.62) LTA4HMAPTNPC1RAB9AHTR1A
SCHEMBL7828732 0.78 HRH3 (0.47) HRH3MAOBHRH1HRH2
SCHEMBL7840842 0.78 HRH3 (0.47) HRH3MAOBHRH1ALDH1A1HRH2
SCHEMBL7839230 0.78 KCNH2 (0.49) HRH3DRD2MAOBHRH1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541200-A Piperidinyl thiacyclic derivatives MERRELL PHARMACEUTICALS INC. (US) 1996-07-30 US disclosed