SCHEMBL9099800

SCHEMBL9099800

CN(C)CCOc1ccc(/C(=C(\CCCl)c2ccccc2)c2ccc(OCc3ccccc3)cc2)cc1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.86
LMNA P02545 2/20 0.86
ESR1 P03372 13/20 0.83
ESRRG P62508 12/20 0.83
ESR2 Q92731 5/20 0.69
MAPT P10636 3/20 0.65
MEN1 O00255 2/20 0.65
TP53 P04637 2/20 0.65
PGR P06401 2/20 0.65
CYP3A4 P08684 2/20 0.65
KMT2A Q03164 2/20 0.65
ESRRA P11474 2/20 0.65
NPC1 O15118 1/20 0.65
NR1I2 O75469 1/20 0.65
PRKD3 O94806 1/20 0.65
ABCB11 O95342 1/20 0.65
EGFR P00533 1/20 0.65
GBA1 P04062 1/20 0.65
NR3C1 P04150 1/20 0.65
ERBB2 P04626 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9097522 1.00 HTR6 (0.86) HTR6LMNAESR1ESRRGESR2
SCHEMBL9097517 1.00 HTR6 (0.86) HTR6LMNAESR1ESRRGESR2
SCHEMBL9097277 0.99 HTR6 (0.84) HTR6LMNAESR1ESRRGESR2
SCHEMBL9097271 0.99 HTR6 (0.84) HTR6LMNAESR1ESRRGESR2
Toremifene SCHEMBL906278 0.93 HTR6 (1.00) HTR6LMNAESR1ESRRGESR2
Toremifene SCHEMBL7465 0.93 HTR6 (1.00) HTR6LMNAESR1ESRRGESR2
Toremifene SCHEMBL1152000 0.93 HTR6 (1.00) HTR6LMNAESR1ESRRGESR2
Toremifene SCHEMBL2223880 0.92 HTR6 (0.97) HTR6LMNAESR1ESRRGESR2
4-Hydroxytormifene SCHEMBL906309 0.91 ESR1 (1.00) HTR6LMNAESR1ESRRGESR2
4-Hydroxytormifene SCHEMBL9099337 0.91 ESR1 (1.00) HTR6LMNAESR1ESRRGESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5491173-A ESTROGENIC, ANTIESTROGENIC AGENTS, ANTITUMOR AGENTS ORION-YHTYMA OY (FI) 1996-02-13 US disclosed