SCHEMBL9102355

SCHEMBL9102355

CCc1ccc(C(=O)N(NC(=O)c2cccc([N+](=O)[O-])c2)C(C)(C)C)c(F)c1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.63
HPGD P15428 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP3A4 P08684 3/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP2C9 P11712 2/20 0.44
CYP1A2 P05177 1/20 0.44
THRA P10827 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5057388 0.92 ABCB1 (0.56) ABCB1HPGDSMN1; SMN2CYP3A4ALDH1A1
SCHEMBL17416592 0.82 ADRB2 (0.42) ABCB1HPGDCYP3A4ALDH1A1LMNA
SCHEMBL9714304 0.81 ABCB1 (0.75) ABCB1HPGDSMN1; SMN2CYP3A4ALDH1A1
SCHEMBL9903862 0.80 HPGD (0.63) ABCB1HPGDSMN1; SMN2CYP3A4
SCHEMBL9714597 0.79 ABCB1 (0.76) ABCB1HPGDSMN1; SMN2CYP3A4ALDH1A1
SCHEMBL5053798 0.78 HPGD (0.43) ABCB1HPGDSMN1; SMN2CYP3A4LMNA
SCHEMBL17416639 0.78 CYP1A2 (0.42) ABCB1HPGDALDH1A1LMNAL3MBTL1
SCHEMBL9101065 0.77 HPGD (0.52) ABCB1HPGDSMN1; SMN2CYP3A4
SCHEMBL5058555 0.77 ABCB1 (0.58) ABCB1HPGDSMN1; SMN2CYP3A4CYP2C9
SCHEMBL9714603 0.77 CYP3A4 (0.73) ABCB1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP disclosed