SCHEMBL9103960

SCHEMBL9103960

O=C(CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1Cc1ccc(F)cc1)NC(Cl)Cc1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.43
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
MEN1 O00255 5/20 0.37
KMT2A Q03164 5/20 0.37
MAPK1 P28482 2/20 0.36
AVPR1A P37288 4/20 0.36
OXTR P30559 1/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9101222 0.90 ITGB2 (0.39) MAPTHDAC1HDAC8HDAC6MEN1
SCHEMBL3700729 0.88 MAPT (0.40) MAPTHDAC1HDAC8HDAC6ITGB2
SCHEMBL9099926 0.85 HDAC1 (0.32) MAPTHDAC1HDAC8HDAC6AVPR1A
SCHEMBL9107165 0.80 MAPT (0.47) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3701041 0.80 MAPT (0.35) MAPTHDAC1HDAC8HDAC6AVPR1A
SCHEMBL9103931 0.80 ITGB2 (0.44) MAPTHDAC1HDAC8HDAC6MEN1
SCHEMBL3704831 0.79 APAF1 (0.36) MAPTHDAC1HDAC8HDAC6AVPR1A
SCHEMBL3705192 0.79 MAPT (0.37) MAPTHDAC1HDAC8HDAC6MEN1
SCHEMBL9102425 0.78 MAPT (0.44) MAPTMEN1KMT2AITGB2ICAM1
SCHEMBL3697542 0.77 ITGB2 (0.40) MAPTHDAC1HDAC8HDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460798-A2 APAF-1 INHIBITOR COMPOUNDS Laboratorios SALVAT, S.A. (ES) 2012-06-06 EP disclosed