SCHEMBL9102425

SCHEMBL9102425

O=C(CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1Cc1ccncc1)NCCc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.38
TRPA1 O75762 1/20 0.38
MDM2 Q00987 1/20 0.38
ITGB2 P05107 1/20 0.38
ICAM1 P05362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9102458 0.97 MAPT (0.42) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL3704087 0.92 TAAR1 (0.44) MAPTALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL9103931 0.88 ITGB2 (0.44) MAPTALDH1A1MEN1KMT2ANPSR1
SCHEMBL3698675 0.88 ALDH1A1 (0.47) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL9105229 0.88 ITGB2 (0.39) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL3700824 0.88 ITGB2 (0.37) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL9101222 0.88 ITGB2 (0.39) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL3698682 0.87 BCHE (0.46) ALDH1A1MEN1KMT2A
SCHEMBL3697146 0.86 KDM4E (0.47) MAPTALDH1A1KDM4ELMNACYP1A2
SCHEMBL3697542 0.86 ITGB2 (0.40) MAPTALDH1A1MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460798-A2 APAF-1 INHIBITOR COMPOUNDS Laboratorios SALVAT, S.A. (ES) 2012-06-06 EP disclosed