SCHEMBL9106413

SCHEMBL9106413

CNC(=O)Nc1ccccc1-c1ccc(CN2C(=O)[C@H](NC(=O)CC(C)(C)NCc3cnco3)CSc3ccccc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.41
XIAP P98170 3/20 0.41
AGTR1 P30556 1/20 0.39
F7 P08709 4/20 0.35
F3 P13726 4/20 0.35
F2 P00734 1/20 0.35
MME P08473 3/20 0.34
ACE P12821 3/20 0.34
RIPK1 Q13546 1/20 0.34
NPY1R P25929 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9104616 0.93 GHSR (0.43) GHSRXIAPAGTR1F7F3
SCHEMBL9108493 0.91 XIAP (0.42) GHSRXIAPAGTR1F7F3
SCHEMBL9108492 0.91 GHSR (0.52) GHSRXIAPAGTR1F7F3
SCHEMBL9107964 0.88 GHSR (0.53) GHSRXIAPAGTR1NPY1R
SCHEMBL9030610 0.87 XIAP (0.42) GHSRXIAPAGTR1F7F3
SCHEMBL9109384 0.86 GHSR (0.40) GHSRXIAPAGTR1F7F3
SCHEMBL9109388 0.86 GHSR (0.40) GHSRXIAPAGTR1F7F3
SCHEMBL9105693 0.85 GHSR (0.44) GHSRXIAPAGTR1F7F3
SCHEMBL7794433 0.85 XIAP (0.47) GHSRXIAPAGTR1F7F3
SCHEMBL7785847 0.84 GHSR (0.51) GHSRXIAPAGTR1F7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430144-A E.g, N-(1-((2'-((methoxycarbonyl)amino)(1,1'-biphenyl)-4-yl) methyl)-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3-yl)-3 ((fur-2-yl)methyl)amino-3-methylbutanamide MERCK & CO., INC. (US) 1995-07-04 US disclosed