SCHEMBL9106773

SCHEMBL9106773

Nc1c2c(nc3cc(C(F)(F)F)ccc13)C1CCC2C1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.66
BCHE P06276 3/20 0.60
CTSD P07339 2/20 0.40
BACE1 P56817 1/20 0.36
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10532976 0.90 ACHE (0.66) ACHEBCHEBACE1CHRNB2CHRNA4
SCHEMBL9104297 0.82 ACHE (0.71) ACHEBCHE
SCHEMBL10468399 0.81 BCHE (0.45) ACHEBCHE
SCHEMBL9107842 0.80 ACHE (1.00) ACHEBCHE
SCHEMBL9107496 0.80 ACHE (0.71) ACHEBCHE
SCHEMBL9105019 0.76 ACHE (0.66) ACHEBCHE
SCHEMBL9106523 0.76 ACHE (1.00) ACHEBCHE
SCHEMBL9597952 0.76 ACHE (0.42) ACHEBCHECTSDBACE1ATM
SCHEMBL9107713 0.75 ACHE (0.41) ACHEBCHE
Hydrochloric Acid SCHEMBL10656143 0.75 ACHE (0.97) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5401749-A Memory enhancers, cholinergic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-03-28 US claimed
US-5401749-A Memory enhancers, cholinergic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-03-28 US disclosed
EP-0278499-B1 9-Amino-1,4-ethano-1,2,3,4-tetrahydroacridine and related compounds, intermediates and a process for the preparation thereof and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1994-09-28 EP disclosed
US-5232927-A Useful for enhancing memory HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-08-03 US disclosed
US-5202440-A Certain 9-amino-2-(or 4)-oxa 1,2,3,4-tetrahydro- or 1,2,3,4,5,6,7,8-octahydro-acridines PFIZER INC. (US) 1993-04-13 US disclosed
US-5037833-A Anticholinergic agents; alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4897400-A ENHANCING MEMORY HOESCHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-01-30 US disclosed
EP-0311303-A2 4-aminopyridine derivatives PFIZER INC. (US) 1989-04-12 EP disclosed
WO-1989002740-A1 4-AMINOPYRIDINE DERIVATIVES PFIZER INC. (US) 1989-04-06 WO disclosed
EP-0306826-A1 N-(substituted alkylidene)fused bicycloalkylidene and hetero-alkylidene quinolinamines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-03-15 EP disclosed
EP-0278499-A2 9-Amino-1,4-ethano-1,2,3,4-tetrahydroacridine and related compounds, intermediates and a process for the preparation thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-08-17 EP disclosed