SCHEMBL911093

SCHEMBL911093

CSc1ccc(OBOc2ccc(SC)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 5/20 0.47
CYP1A2 P05177 5/20 0.47
CYP1B1 Q16678 5/20 0.47
ALDH1A1 P00352 2/20 0.39
SLC6A4 P31645 5/20 0.37
MAOB P27338 1/20 0.37
AOC3 Q16853 1/20 0.37
HTR2A P28223 1/20 0.37
KCNH2 Q12809 1/20 0.37
GAA P10253 1/20 0.37
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
PLK1 P53350 1/20 0.34
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15257351 0.81 CYP1A1 (0.44) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
SCHEMBL2774995 0.76 CYP1A1 (0.52) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
SCHEMBL4017550 0.75 AR (0.36) CYP1A2ALDH1A1SLC6A4KCNH2
SCHEMBL4520712 0.75 SLC6A4 (0.41) CYP1A2ALDH1A1SLC6A4MAOBMAOA
SCHEMBL83839 0.74 ALDH1A1 (0.58) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
SCHEMBL1145983 0.74 CYP1A1 (0.75) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
SCHEMBL11986269 0.74 CYP1A1 (0.75) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
SCHEMBL4040069 0.73 SMN1; SMN2 (0.39) CYP1A1CYP1A2CYP1B1ALDH1A1GAA
SCHEMBL1146090 0.72 CYP1A1 (0.48) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4
Hydrogen Sulfide SCHEMBL17008164 0.72 CYP1A1 (0.72) CYP1A1CYP1A2CYP1B1ALDH1A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023027630-A9 A FLOW REACTOR, METHODS OF FABRICATION AND REACTIONS THEREOF NATIONAL UNIVERSITY OF SINGAPORE (SG) 2023-07-27 WO claimed
WO-2023027630-A2 A FLOW REACTOR, METHODS OF FABRICATION AND REACTIONS THEREOF NATIONAL UNIVERSITY OF SINGAPORE (SG) 2023-03-02 WO claimed
US-8921299-B2 Detergents having acceptable color THE PROCTER & GAMBLE COMPANY (US) 2014-12-30 US claimed
WO-2023027630-A9 A FLOW REACTOR, METHODS OF FABRICATION AND REACTIONS THEREOF NATIONAL UNIVERSITY OF SINGAPORE (SG) 2023-07-27 WO disclosed
WO-2023027630-A2 A FLOW REACTOR, METHODS OF FABRICATION AND REACTIONS THEREOF NATIONAL UNIVERSITY OF SINGAPORE (SG) 2023-03-02 WO disclosed
US-20210171865-A1 Detergent Composition Arxada, LLC 2021-06-10 US disclosed
EP-1613613-B1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORP (US) 2021-06-02 EP disclosed
EP-3823584-A1 DETERGENT COMPOSITION LONZA, LLC (US) 2021-05-26 EP disclosed
WO-2020018891-A1 DETERGENT COMPOSITION LONZA INC. (US) 2020-01-23 WO disclosed
EP-3191465-B1 HERBICIDAL QUINOLINES SYNGENTA PARTICIPATIONS AG (CH) 2018-12-19 EP disclosed
US-9980486-B2 Herbicidal quinolines SYNGENTA PARTICIPATIONS AG (CH) 2018-05-29 US disclosed
EP-0853083-B1 Pyridylfuran and pyridylthiophene compounds and pharmaceutical use thereof PFIZER (US) 2001-09-12 EP disclosed
EP-1015431-A1 2-AMINOPYRIDINES AS INHIBITORS OF CYCLOOXYGENASE-2 Merck Frosst Canada & Co. (CA) 2000-07-05 EP disclosed
US-6048880-A THERAPY FOR CYTOKINE SENSITIVE DISEASES PFIZER PHARAMACEUTICALS INC. (JP) 2000-04-11 US disclosed
EP-0975604-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 Merck Frosst Canada & Co. (CA) 2000-02-02 EP disclosed
US-6004950-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; ANALGESIC, ANTIPYRETICS; SIDE EFFECT REDUCTION MERCK FROSST CANADA, INC. (CA) 1999-12-21 US disclosed
US-6004960-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION MERCK FROSST CANADA, INC. (CA) 1999-12-21 US disclosed
WO-1999014195-A1 2-AMINOPYRIDINES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 1999-03-25 WO disclosed
WO-1998041511-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 1998-09-24 WO disclosed
EP-0853083-A1 Pyridylfuran and pyridylthiophene compounds and pharmaceutical use thereof PFIZER INC. (US) 1998-07-15 EP disclosed