SCHEMBL9112199

SCHEMBL9112199

Nc1cc(N)c(C[O])c(N)c1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TSHR P16473 2/20 0.32
PTK2 Q05397 1/20 0.32
CASP1 P29466 1/20 0.31
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9112204 0.71 KDM4E (0.33) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL27941110 0.71 TSHR (0.43) TDP1ALDH1A1TSHRCASP1CYP3A4
SCHEMBL10432144 0.69 DHFR (0.36) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL1002823 0.69 KDM4E (0.42) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL18421930 0.67 KDM4E (0.31) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL16869681 0.65 KDM4E (0.34) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL27770925 0.65 CASP1 (0.42) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL293508 0.65 PTK2 (0.38) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL4284421 0.63 CYP3A4 (0.44) TDP1KDM4EMEN1KMT2AALDH1A1
SCHEMBL7350411 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1114834-A antidiabetic agent OTSUKA PHARMA CO LTD (JP) 1996-01-10 CN disclosed
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed