SCHEMBL9112952

SCHEMBL9112952

O=C(Nc1ccccc1)Nc1nnnn1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.52
TSHR P16473 2/20 0.52
TP53 P04637 2/20 0.52
EPHX1 P07099 1/20 0.52
EPHX2 P34913 1/20 0.52
CDK9 P50750 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
KCNJ6 P48051 1/20 0.51
KCNJ5 P48544 1/20 0.51
KCNJ3 P48549 1/20 0.51
ALDH1A1 P00352 4/20 0.50
ADORA3 P0DMS8 2/20 0.50
HTT P42858 2/20 0.50
LMNA P02545 1/20 0.50
MAPK13 O15264 3/20 0.49
MAPK12 P53778 3/20 0.49
MAPK11 Q15759 3/20 0.49
MAPK14 Q16539 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
CYP1A2 P05177 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17533119 0.83 MAPK1 (0.58) SMN1; SMN2ALDH1A1ADORA3HTTLMNA
SCHEMBL4772885 0.80 POLB (0.59) SMN1; SMN2TSHRTP53EPHX1EPHX2
SCHEMBL14498671 0.79 TSHR (0.49) SMN1; SMN2TSHRTP53EPHX1EPHX2
SCHEMBL7346662 0.78 ALDH1A1 (0.55) SMN1; SMN2TSHRALDH1A1HTTLMNA
SCHEMBL8507647 0.77 GAA (0.59) SMN1; SMN2TSHRALDH1A1HTTLMNA
SCHEMBL14498648 0.76 TSHR (0.46) SMN1; SMN2TSHRTP53EPHX1EPHX2
SCHEMBL18292654 0.75 GAA (0.64) SMN1; SMN2TSHRALDH1A1HTTLMNA
Diphenylurea SCHEMBL133103 0.72 SMN1; SMN2 (1.00) SMN1; SMN2TSHRTP53EPHX1EPHX2
SCHEMBL14590428 0.72 ALDH1A1 (0.60) SMN1; SMN2TSHRALDH1A1HTTLMNA
SCHEMBL14937204 0.72 ALDH1A1 (0.60) SMN1; SMN2TSHRALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995014679-A1 TETRAZOLE-SUBSTITUTED UREA ACAT INHIBITORS PARKE, DAVIS & COMPANY (US) 1995-06-01 WO disclosed
US-5362744-A Treatnent of athrosclerosis, anticholesterol agents WARNER-LAMBERT COMPANY (US) 1994-11-08 US disclosed
US-5073565-A Atherosclerosis, anticholesterol WARNER-LAMBERT COMPANY (US) 1991-12-17 US disclosed
WO-1991017150-A1 TETRAZOLE UREA AND THIOUREA ACAT INHIBITORS WARNER-LAMBERT COMPANY (US) 1991-11-14 WO disclosed