SCHEMBL9113250

SCHEMBL9113250

CCOC(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
MAPT P10636 1/20 0.49
ALDH1A1 P00352 4/20 0.49
TGM2 P21980 5/20 0.47
AKR1B1 P15121 1/20 0.47
MAPK1 P28482 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
HCRTR1 O43613 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11430193 0.99 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL23577870 0.88 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL22380701 0.83 PDPK1 (0.57) CA12CA1CA2CA7CA9
SCHEMBL30901337 0.82 IDO1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL2241739 0.80 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL7417096 0.79 AKR1B1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL5846673 0.78 MAPT (0.68) CA12CA1CA2CA7CA9
SCHEMBL12273071 0.77 TGM2 (0.56) ALDH1A1TGM2IDO1TDO2CES1
SCHEMBL1680517 0.77 CA12 (0.48) CA12CA1CA2CA7CA9
SCHEMBL1050601 0.76 SMYD3 (0.56) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4186132-A Isatin products THE REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1980-01-29 US claimed
US-5441955-A Tuberculosis PATHOGENESIS CORPORATION (US) 1995-08-15 US disclosed
WO-1995013807-A1 INDOLO[2,1-b]QUINAZOLINE-6,12-DIONE ANTIBACTERIAL COMPOUNDS AND METHODS OF USE THEREOF PATHOGENESIS CORPORATION (US) 1995-05-26 WO disclosed
US-4252723-A Air oxidation of oxindoles to isatins REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1981-02-24 US disclosed
US-4188325-A Isatin process and products REGENTS OF UNIVERSITY OF MINNESOTA (US) 1980-02-12 US disclosed
US-4186132-A Isatin products THE REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1980-01-29 US disclosed