SCHEMBL9113592

SCHEMBL9113592

[CH2]C=CC(=O)N(CC)CCC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.40
CA9 Q16790 4/20 0.40
CA2 P00918 3/20 0.40
CYP3A4 P08684 1/20 0.40
NPC1 O15118 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
APP P05067 2/20 0.36
CA1 P00915 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9113596 0.81 CA12 (0.41) CA12CA9CA2CYP3A4NPC1
SCHEMBL19854404 0.79 ZDHHC20 (0.50) CA12CA9CA2CYP3A4NPC1
SCHEMBL19917777 0.79 ZDHHC20 (0.50) CA12CA9CA2CYP3A4NPC1
SCHEMBL2560026 0.78 ZDHHC20 (0.47) CA12CA9CA2CYP3A4NPC1
SCHEMBL1834006 0.77 CA12 (0.50) CA12CA9CA2CYP3A4NPC1
SCHEMBL9070448 0.75 CYP3A4 (0.37) CA12CA9CA2CYP3A4NPC1
SCHEMBL3468531 0.72 CA12 (0.50) CA12CA9CA2TSHRMAPK1
SCHEMBL12924014 0.72 PPARG (0.46) CYP3A4TP53LMNAMMP2
SCHEMBL1022195 0.71 NPC1 (0.54) CA12CA9CA2CYP3A4NPC1
SCHEMBL1395649 0.71 NPC1 (0.54) CA12CA9CA2CYP3A4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1114834-A antidiabetic agent OTSUKA PHARMA CO LTD (JP) 1996-01-10 CN disclosed
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed