SCHEMBL9114098

SCHEMBL9114098

[CH2]C=CCCCc1nccc2occc12

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.33
HTR2C P28335 1/20 0.33
DRD1 P21728 1/20 0.30
FADS1 O60427 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9112011 0.81 HTR2C (0.36) TRPA1HTR2CDRD1FADS1
SCHEMBL9109755 0.78 HTR2C (0.33) TRPA1HTR2CDRD1FADS1
SCHEMBL9113672 0.75 HTR2C (0.33) TRPA1HTR2CFADS1
SCHEMBL9113007 0.73 TRPA1 (0.33) TRPA1HTR2CDRD1FADS1
SCHEMBL9112969 0.73 HTR2C (0.34) TRPA1HTR2CDRD1FADS1
SCHEMBL9113177 0.69 HTR2C (0.33) TRPA1HTR2CDRD1FADS1
SCHEMBL9113881 0.69 CHRM2 (0.52)
SCHEMBL3803166 0.69 HTR2C (0.40) TRPA1HTR2CDRD1FADS1
SCHEMBL31426315 0.69 PDE3B (0.42) TRPA1HTR2CDRD1FADS1
SCHEMBL8371407 0.69 HTR2C (0.42) TRPA1HTR2CDRD1FADS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed