SCHEMBL9115680

SCHEMBL9115680

COc1cc2occ(CCCN3CCC(C(=O)c4ccc(F)cc4)CC3)c(=O)c2cc1OC

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.49
HTR2C P28335 2/20 0.49
DRD2 P14416 1/20 0.49
CYP2D6 P10635 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HTR7 P34969 1/20 0.48
HTR6 P50406 1/20 0.48
WNT3A P56704 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9115270 0.97 HTR2A (0.52) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9118367 0.97 HTR2A (0.51) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9115669 0.97 HTR2A (0.51) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9116119 0.97 HTR2A (0.51) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9115389 0.92 MAPT (0.45) MAPTSMN1; SMN2
SCHEMBL9117021 0.91 KCNH2 (0.48) HTR2ACYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL9116840 0.89 KCNH2 (0.45) HTR2AHTR2CDRD2HTR7
SCHEMBL9114665 0.89 DRD2 (0.49) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9116078 0.86 HTR2A (0.51) HTR2AHTR2CDRD2CYP2D6KDM4E
SCHEMBL9118626 0.86 HTR2A (0.50) HTR2AHTR2CCYP2D6KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO claimed