SCHEMBL9116840

SCHEMBL9116840

COc1cc2occ(CCCN3CCC(C(=O)c4ccc(F)cc4F)CC3)c(=O)c2cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.45
HTR2A P28223 5/20 0.44
GRM2 Q14416 3/20 0.44
DRD4 P21917 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
DRD3 P35462 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
PDE10A Q9Y233 2/20 0.40
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2C P18825 1/20 0.39
DRD1 P21728 1/20 0.39
DRD5 P21918 1/20 0.39
HRH2 P25021 1/20 0.39
HTR1D P28221 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117345 0.89 CHRM2 (0.49) KCNH2DRD4CHRM2CHRM4CHRM5
SCHEMBL9115680 0.89 HTR2A (0.49) HTR2ADRD2HTR2CHTR7
SCHEMBL9115270 0.87 HTR2A (0.52) HTR2ADRD2HTR2CHTR7
SCHEMBL9116119 0.86 HTR2A (0.51) HTR2ADRD2HTR2CHTR7
SCHEMBL9115669 0.86 HTR2A (0.51) HTR2ADRD2HTR2CHTR7
SCHEMBL9118367 0.86 HTR2A (0.51) HTR2ADRD2HTR2CHTR7
SCHEMBL9116097 0.85 ALDH1A1 (0.51) KCNH2HTR2ADRD4CHRM2CHRM4
SCHEMBL9117021 0.84 KCNH2 (0.48) KCNH2HTR2A
SCHEMBL9115389 0.83 MAPT (0.45) KCNH2
SCHEMBL9114665 0.78 DRD2 (0.49) HTR2ADRD2HTR2CHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO claimed
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO disclosed