SCHEMBL9116053

SCHEMBL9116053

COc1cc(CCC(=O)N(C)CC(c2ccccc2)c2ccccc2)cc(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.62
TDP1 Q9NUW8 1/20 0.50
KMT2A Q03164 3/20 0.47
CCR5 P51681 1/20 0.46
DUT P33316 1/20 0.46
MEN1 O00255 2/20 0.44
GAA P10253 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HIF1A Q16665 1/20 0.41
FFAR1 O14842 1/20 0.41
NR1H3 Q13133 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9239998 0.88 TACR1 (0.59) TACR1TDP1KMT2ACCR5MEN1
SCHEMBL9114494 0.87 TACR1 (0.64) TACR1TDP1KMT2ACCR5MEN1
SCHEMBL9114531 0.80 TACR1 (0.77) TACR1TDP1KMT2ACCR5MEN1
SCHEMBL9112802 0.79 TACR1 (0.61) TACR1TDP1KMT2AMEN1NPC1
SCHEMBL9114442 0.76 TACR1 (1.00) TACR1TDP1KMT2ACCR5MEN1
SCHEMBL9114227 0.75 TACR1 (0.61) TACR1KMT2AMEN1GAARAB9A
SCHEMBL9114068 0.75 TACR1 (0.64) TACR1TDP1KMT2AMEN1
SCHEMBL9114062 0.74 TACR1 (0.62) TACR1TDP1KMT2ACCR5MEN1
SCHEMBL9117035 0.73 MTNR1A (0.65) TACR1KMT2AMEN1GAAPOLB
SCHEMBL7194988 0.73 NPC1 (0.69) TDP1KMT2AMEN1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995011880-A1 SUBSTITUTED AMIDES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-05-04 WO disclosed