SCHEMBL9116873

SCHEMBL9116873

COc1ccc2cc([C@@H](C)C(=O)O)ccc2c1Br

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 16/20 0.58
AKR1C2 P52895 16/20 0.58
PTGS2 P35354 3/20 0.58
PTGS1 P23219 2/20 0.58
CDC42 P60953 1/20 0.58
RAC1 P63000 1/20 0.58
CYP1A2 P05177 1/20 0.58
TSHR P16473 1/20 0.58
SLC22A6 Q4U2R8 1/20 0.58
AKR1B1 P15121 1/20 0.53
LMNA P02545 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4380164 1.00 AKR1C3 (0.58) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL4380166 1.00 AKR1C3 (0.58) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL9239300 0.88 RXFP1 (0.47) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL7772358 0.88 PTGS2 (0.45) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL9243634 0.88 RXFP1 (0.44) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL10537008 0.88 RXFP1 (0.47) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL9868774 0.85 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL9868769 0.85 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2PTGS1CDC42
SCHEMBL9868760 0.85 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2PTGS1CDC42
Methoxymethane SCHEMBL10539889 0.84 AKR1C3 (0.42) AKR1C3AKR1C2PTGS2PTGS1CDC42

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0398288-B1 Process for preparing optically active 2-arylalkanoic acids, in particular 2-arylpropionic acids PUETTER MEDICE CHEM PHARM (DE) 1995-10-18 EP disclosed
US-5380927-A Process for preparing optically active 2-aryl-alkanoic acids, in particular 2-aryl-propionic acids MEDICE CHEM.-PHARM. FABRIK PUTTER GMBH & CO. KG (DE) 1995-01-10 US disclosed
US-5266723-A Process for the preparation of optically active 2-aryl-alkanoic acids, especially 2-aryl-propionic acids MEDICE, LTD., CHEM.-PHARM. FABRIK PUTTER GMBH & CO. KG (DE) 1993-11-30 US disclosed
US-4888433-A CHIRAL HALOGENATED KETALS WHICH UNDERGO STEREOSELECTIVE REARRANGEMENT ZAMBON, S.P.A. (IT) 1989-12-19 US disclosed
US-4810819-A STEREOSELECTIVE HALOGENATION AND REARRANGEMENT ZAMBON SPA (IT) 1989-03-07 US disclosed
EP-0158913-B1 PROCESS FOR THE PREPARATION OF OPTICALLY ACTIVE ALPHA-ARYLALKANOIC ACIDS AND INTERMEDIATES THEREOF ZAMBON S.p.A. (IT) 1988-07-20 EP disclosed
US-4697036-A HALOGENATION, REARRANGEMENT ZAMBON S.P.A. (IT) 1987-09-29 US disclosed
EP-0158913-A2 Process for the preparation of optically active alpha-arylalkanoic acids and intermediates thereof ZAMBON S.p.A. (IT) 1985-10-23 EP disclosed