SCHEMBL9116909

SCHEMBL9116909

CC(O)(C#CBr)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
CYP2C19 P33261 3/20 0.40
CYP2D6 P10635 2/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 2/20 0.38
KMT2A Q03164 2/20 0.38
PABPC1 P11940 1/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
MAPT P10636 1/20 0.38
HIF1A Q16665 1/20 0.36
MEN1 O00255 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
CYP2B6 P20813 1/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017366 0.86 ALDH1A1 (0.46) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL10271603 0.80 ALDH1A1 (0.41) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL15165102 0.79 ALDH1A1 (0.42) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL172920 0.78 ALDH1A1 (0.40) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL9114456 0.78 ALDH1A1 (0.40) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL31261832 0.77 KDM4E (0.47) ALDH1A1CYP2C19CYP2D6HSD17B10KDM4E
SCHEMBL523695 0.77 MAPT (0.51) ALDH1A1CYP2C19ALOX15ESR1ESR2
SCHEMBL28397568 0.75 ALDH1A1 (0.38) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL9806921 0.75 ALDH1A1 (0.42) ALDH1A1CYP2C19CYP2D6ALOX15HSD17B10
SCHEMBL127044 0.73 ALDH1A1 (0.43) ALDH1A1CYP2C19ALOX15ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446203-A Synthesis of haloenones and aryl or alkyl substituted enones or alkenes NEW YORK UNIVERSITY (US) 1995-08-29 US disclosed
EP-0656878-A4 SYNTHESIS OF HALOENONES AND ARYL OR ALKYL SUBSTITUTED ENONES OR ALKENES. 1995-07-05 EP disclosed
EP-0656878-A1 SYNTHESIS OF HALOENONES AND ARYL OR ALKYL SUBSTITUTED ENONES OR ALKENES NEW YORK UNIVERSITY (US) 1995-06-14 EP disclosed
WO-1994005617-A1 SYNTHESIS OF HALOENONES AND ARYL OR ALKYL SUBSTITUTED ENONES OR ALKENES NEW YORK UNIVERSITY (US) 1994-03-17 WO disclosed