SCHEMBL9117151

SCHEMBL9117151

NS(=O)(=O)c1ccc(C2=CC3(C=C2c2ccc(C(F)(F)F)cc2)CCC3)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.47
PTGS2 P35354 8/20 0.46
PTGS1 P23219 3/20 0.46
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
CA4 P22748 2/20 0.38
CA7 P43166 2/20 0.38
PDPK1 O15530 1/20 0.37
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
KDM1A O60341 1/20 0.36
MAOB P27338 1/20 0.36
GCK P35557 1/20 0.36
GCKR Q14397 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117239 0.98 KIF11 (0.47) KIF11PTGS2PTGS1KDM4EGAA
SCHEMBL9235736 0.95 KIF11 (0.49) KIF11PTGS2PTGS1KDM4EGAA
SCHEMBL9119018 0.93 KIF11 (0.47) KIF11PTGS2PTGS1KDM4ECYP2C9
SCHEMBL9118931 0.91 KIF11 (0.47) KIF11PTGS2PTGS1KDM4ECYP2C9
SCHEMBL9118118 0.89 KIF11 (0.49) KIF11PTGS2PTGS1CYP2C9CA12
SCHEMBL9117334 0.87 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973751 0.87 KIF11 (0.52) KIF11PTGS2PTGS1KDM4EGAA
SCHEMBL9118443 0.87 KIF11 (0.62) KIF11PTGS2PTGS1CYP2C9CA12
SCHEMBL9115739 0.87 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8974399 0.85 KIF11 (0.50) KIF11PTGS2PTGS1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed