SCHEMBL9117293

SCHEMBL9117293

COc1ccc2occ(CCCN3CCC(C(=O)c4ccc(NS(C)(=O)=O)cc4)CC3)c(=O)c2c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
POLB P06746 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MTNR1A P48039 7/20 0.45
MTNR1B P49286 3/20 0.45
MAOB P27338 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
NQO2 P16083 1/20 0.41
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALDH2 P05091 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9114665 0.87 DRD2 (0.49) CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL9116820 0.87 MAOB (0.51) KCNH2KDM4EMTNR1AMTNR1BMAOB
SCHEMBL9115835 0.84 HTR2A (0.50) CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL9115981 0.84 HTR2A (0.50) CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL9115963 0.84 HTR2A (0.50) CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL9115389 0.82 MAPT (0.45) KCNH2POLBTDP1ALDH1A1
SCHEMBL9117585 0.82 HTR2A (0.51) CYP2C19ALDH1A1
SCHEMBL9117040 0.81 MAOB (0.51) KCNH2CYP3A4KDM4EMAOBALDH1A1
SCHEMBL9116972 0.80 DRD2 (0.47) CYP3A4CYP2D6KDM4E
SCHEMBL9116078 0.79 HTR2A (0.51) CYP3A4CYP2D6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO disclosed