SCHEMBL9117936

SCHEMBL9117936

CS(=O)(=O)c1ccc(C2=CC(CF)(CF)C=C2c2ccc(Cl)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.55
PTGS1 P23219 6/20 0.50
RORC P51449 1/20 0.46
DRD1 P21728 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974351 0.86 PTGS2 (0.57) PTGS2PTGS1RORC
SCHEMBL8974299 0.86 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8974954 0.85 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL8974391 0.85 PTGS2 (0.59) PTGS2PTGS1RORC
SCHEMBL8974098 0.84 PTGS2 (0.48) PTGS2PTGS1DRD1
SCHEMBL8974128 0.83 PTGS2 (0.56) PTGS2PTGS1RORC
SCHEMBL9117490 0.82 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8974669 0.81 PTGS2 (0.59) PTGS2PTGS1RORC
SCHEMBL8974363 0.79 PTGS2 (0.47) PTGS2PTGS1DRD1
SCHEMBL8975150 0.79 PTGS2 (0.51) PTGS2PTGS1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed