SCHEMBL9118050

SCHEMBL9118050

Oc1cccc2c1CC[C@@H]1[C@H]2CCN1CCC1CCCCC1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.70
HTR1A P08908 8/20 0.70
CHRM2 P08172 1/20 0.64
CHRM1 P11229 1/20 0.64
CHRM3 P20309 1/20 0.64
ACHE P22303 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118057 1.00 DRD2 (0.70) DRD2HTR1ACHRM2CHRM1CHRM3
Hydrochloric Acid SCHEMBL9441210 0.99 DRD2 (0.69) DRD2HTR1ACHRM2CHRM1CHRM3
Hydrochloric Acid SCHEMBL9118521 0.99 DRD2 (0.69) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9121632 0.99 DRD2 (0.72) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9121623 0.99 DRD2 (0.72) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9119644 0.93 DRD2 (0.67) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9119638 0.93 DRD2 (0.67) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9117994 0.92 DRD2 (0.66) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9117991 0.92 DRD2 (0.66) DRD2HTR1ACHRM2CHRM1CHRM3
SCHEMBL9121991 0.92 DRD2 (0.69) DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548664-B1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives HOFFMANN LA ROCHE (CH) 1995-05-31 EP disclosed
US-5318966-A Administering the enzyme inhibitor for treating alzheimer's disease, learning enhancement, brain disorders HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
US-5318967-A Cognition activators for alzheimer's disease, learning enhancement HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
EP-0548664-A1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed