SCHEMBL9118085

SCHEMBL9118085

CS(=O)(=O)c1ccc(C2=CC3(C=C2c2ccccc2)CCCC3)nc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.48
PTGS1 P23219 5/20 0.48
RORC P51449 2/20 0.40
OPRL1 P41146 1/20 0.37
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118010 0.97 PTGS2 (0.48) PTGS2PTGS1RORCOPRL1JAK2
SCHEMBL9115482 0.95 PTGS2 (0.53) PTGS2PTGS1RORCOPRL1JAK2
SCHEMBL9242947 0.89 PTGS2 (0.50) PTGS2PTGS1RORC
SCHEMBL9117188 0.88 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL9118366 0.88 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL9116102 0.88 CA2 (0.40) PTGS2PTGS1
SCHEMBL9117225 0.86 PTGS2 (0.50) PTGS2PTGS1RORC
SCHEMBL9118519 0.86 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL9242413 0.86 PTGS2 (0.47) PTGS2PTGS1RORC
SCHEMBL9118717 0.85 PTGS2 (0.49) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed