SCHEMBL9118751

SCHEMBL9118751

COc1ccc(C2=CC3(C=C2c2ccc(S(=O)(=O)CF)cc2)CC3)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.59
PTGS1 P23219 4/20 0.59
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
PDE4B Q07343 2/20 0.37
PDE4D Q08499 2/20 0.37
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
KMT2A Q03164 1/20 0.36
PAX8 Q06710 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
CYP19A1 P11511 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118171 0.91 PTGS2 (0.57) PTGS2PTGS1POLBTSHRKMT2A
SCHEMBL9117634 0.91 PTGS2 (0.57) PTGS2PTGS1TSHRMAPK1MAPT
SCHEMBL9117521 0.91 PTGS2 (0.57) PTGS2PTGS1KMT2A
SCHEMBL9117087 0.90 PTGS2 (0.75) PTGS2PTGS1
SCHEMBL9117671 0.89 PTGS2 (0.52) PTGS2PTGS1POLBKMT2AMAPT
SCHEMBL9118113 0.85 PTGS2 (0.79) PTGS2PTGS1POLBTSHRMAPK1
SCHEMBL9116418 0.84 PTGS2 (0.60) PTGS2PTGS1POLBTSHRMAPK1
SCHEMBL9116116 0.84 PTGS2 (0.62) PTGS2PTGS1MAPK1KMT2AMAPT
SCHEMBL9116863 0.83 PTGS2 (0.59) PTGS2PTGS1POLBTSHRMAPK1
SCHEMBL9117086 0.82 PTGS2 (0.46) PTGS2PTGS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed