SCHEMBL9119210

SCHEMBL9119210

C=CC[C@H](C(=O)N(C)Cc1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
SLC6A4 P31645 2/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
HSP90AA1 P07900 1/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
ATM Q13315 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801314 0.89 HPGD (0.45) HPGDSLC6A4CA12CA9HSP90AA1
SCHEMBL8801310 0.89 HPGD (0.45) HPGDSLC6A4CA12CA9HSP90AA1
SCHEMBL8691676 0.81 TACR2 (0.44) SLC6A4CYP2C19CYP3A4CYP2D6SLC6A2
SCHEMBL8062847 0.78 SLC6A3 (0.40) SLC6A4CYP2C19LMNACYP3A4CYP2D6
SCHEMBL8062852 0.78 SLC6A3 (0.40) SLC6A4CYP2C19LMNACYP3A4CYP2D6
SCHEMBL624052 0.77 CYP2C19 (0.60) SLC6A4CYP2C19LMNASLC6A2SLC6A3
SCHEMBL5879212 0.77 CYP2C19 (0.60) SLC6A4CYP2C19LMNASLC6A2SLC6A3
SCHEMBL5879216 0.77 CYP2C19 (0.60) SLC6A4CYP2C19LMNASLC6A2SLC6A3
SCHEMBL8689932 0.76 TACR2 (0.42) CYP2C19MEN1KMT2ALMNACYP3A4
SCHEMBL8802198 0.76 TACR3 (0.53) SLC6A4SLC6A2SLC6A3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995028931-A1 SPIRO-SUBSTITUTED AZACYCLES AS NEUROKININ-3 ANTAGONISTS MERCK & CO., INC. (US) 1995-11-02 WO disclosed
US-5434158-A Asthma MERCK & CO., INC. (US) 1995-07-18 US disclosed