SCHEMBL9119310

SCHEMBL9119310

COc1cc(C(=O)N(Cc2ccccc2)C(C)C)ccc1OCCCCCOc1cccc(C(=N)N)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 2/20 0.61
LTB4R2 Q9NPC1 1/20 0.59
PRSS1 P07477 10/20 0.53
NR1H3 Q13133 1/20 0.50
REN P00797 5/20 0.48
F10 P00742 1/20 0.47
HTR1A P08908 2/20 0.47
ADRA1D P25100 2/20 0.47
HTR2A P28223 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
HTR2B P41595 2/20 0.47
KCNH2 Q12809 2/20 0.47
F2 P00734 1/20 0.47
PLG P00747 1/20 0.47
PRSS2 P07478 1/20 0.47
C1S P09871 1/20 0.47
PRSS3 P35030 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118827 0.92 LTB4R (0.73) LTB4RLTB4R2PRSS1RENHTR1A
Hydrochloric Acid SCHEMBL8994911 0.91 LTB4R (0.72) LTB4RLTB4R2PRSS1RENHTR1A
SCHEMBL9119317 0.84 LTB4R (0.48) LTB4RLTB4R2NR1H3RENHTR1A
SCHEMBL8995067 0.83 LTB4R (0.57) LTB4RLTB4R2RENHTR1AADRA1D
SCHEMBL9118833 0.80 LTB4R (0.54) LTB4RLTB4R2RENHTR1AADRA1D
Hydrochloric Acid SCHEMBL8994925 0.80 LTB4R (0.53) LTB4RLTB4R2RENHTR1AADRA1D
Hydrochloric Acid SCHEMBL8994844 0.79 LTB4R (0.67) LTB4RLTB4R2PRSS1F2
Moxilubant SCHEMBL6439215 0.77 LTB4R (1.00) LTB4RLTB4R2PRSS1F10HTR2A
Moxilubant SCHEMBL29388138 0.77 LTB4R (1.00) LTB4RLTB4R2PRSS1F10HTR2A
Moxilubant SCHEMBL8994884 0.76 LTB4R (0.98) LTB4RLTB4R2PRSS1F10HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0518819-B1 Amidino compounds, their manufacture and use as medicament CIBA GEIGY AG (CH) 1995-08-02 EP claimed