SCHEMBL9119782

SCHEMBL9119782

COC(=O)c1cccnc1-c1ccccc1CO

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
PKM P14618 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAP2K1 Q02750 1/20 0.46
ALDH1A1 P00352 3/20 0.45
BDKRB1 P46663 4/20 0.45
KDM4E B2RXH2 4/20 0.45
SLC6A3 Q01959 3/20 0.44
SLC6A4 P31645 2/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 2/20 0.43
ATM Q13315 1/20 0.43
KCNA5 P22460 1/20 0.43
FAAH O00519 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
MAPK10 P53779 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118970 0.88 TDP1 (0.47) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL9301375 0.81 SLC6A3 (0.57) ALDH1A1KDM4ESLC6A3SLC6A4LMNA
SCHEMBL16547421 0.80 TDP1 (0.50) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL22717702 0.80 SLC6A4 (0.50) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL22717355 0.80 KMT2A (0.50) TDP1PKML3MBTL1ALDH1A1KDM4E
SCHEMBL29575477 0.80 KMT2A (0.50) TDP1PKML3MBTL1ALDH1A1KDM4E
SCHEMBL29574044 0.80 SLC6A4 (0.50) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL812065 0.80 KDM4E (0.59) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL7362874 0.77 KDM4E (0.50) TDP1PKML3MBTL1MAP2K1ALDH1A1
SCHEMBL7367740 0.77 KDM4E (0.47) TDP1PKML3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5451583-A Angiotensin inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1995-09-19 US disclosed
WO-1994011365-A1 SUBSTITUTED BENZIMIDAZOLES AND QUINAZOLINES AS ANTIHYPERTENSIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1994-05-26 WO disclosed
US-5283242-A Hypotensive agents, cardiotonic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1994-02-01 US disclosed