SCHEMBL9119818

SCHEMBL9119818

COC(=O)CCCCOc1ccc(OCCCCCOS(C)(=O)=O)c(CCC(=O)OC)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
P2RY12 Q9H244 3/20 0.43
PPARG P37231 4/20 0.42
PPARA Q07869 3/20 0.42
PPARD Q03181 3/20 0.42
MAPT P10636 1/20 0.42
MTNR1B P49286 3/20 0.41
MTNR1A P48039 2/20 0.41
PDE2A O00408 1/20 0.40
LTB4R Q15722 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC1 Q13547 1/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799495 0.89 MEN1 (0.48) PDE3BPDE3AP2RY12PPARGPPARA
SCHEMBL8800390 0.88 LTB4R (0.41) PDE3BPDE3AP2RY12PPARGPPARA
SCHEMBL9117669 0.87 BRD4 (0.45) PDE3BPDE3AP2RY12MEN1KMT2A
SCHEMBL8799721 0.87 MEN1 (0.43) PDE3BPDE3AP2RY12MTNR1BMTNR1A
SCHEMBL9121185 0.86 MAPT (0.41) PPARGPPARAPPARDMAPTMTNR1B
SCHEMBL9121261 0.86 PDE3B (0.46) PDE3BPDE3AP2RY12PPARGPPARA
SCHEMBL9118524 0.84 LTB4R (0.43) MAPTLTB4RMEN1ALDH1A1KMT2A
SCHEMBL9121437 0.83 LTB4R (0.44) PPARGPPARAPPARDMAPTLTB4R
SCHEMBL9121426 0.82 PPARD (0.49) PPARGPPARDLTB4RMEN1ALDH1A1
SCHEMBL8800245 0.82 LTB4R (0.42) PPARGPPARAMAPTLTB4RMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434186-A Antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1995-07-18 US disclosed
US-5273999-A A 4-keto-boroalkyleneoxychroman or 2,3-dihydrobenzofuran derivative HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0531823-A1 Bicyclic carboxylic acid derivatives as anti-inflammatory agents F. HOFFMANN-LA ROCHE AG (CH) 1993-03-17 EP disclosed