SCHEMBL9119829

SCHEMBL9119829

CC(C)(C)c1nc(-c2n[nH]c(=S)s2)nc(C(C)(C)C)c1O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.54
PTGS1 P23219 5/20 0.54
ALOX5 P09917 2/20 0.54
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GAA P10253 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9120355 0.71 PTGS2 (0.40) PTGS2PTGS1ALOX5
SCHEMBL9738587 0.70 PTGS1 (0.40) PTGS2PTGS1ALOX5
SCHEMBL2694570 0.70 PTGS2 (1.00) PTGS2PTGS1ALOX5CA1CA2
SCHEMBL9182983 0.69 PTGS2 (0.97) PTGS2PTGS1ALOX5CA1CA2
SCHEMBL9122434 0.68 PTGS2 (0.54) PTGS2PTGS1KDM4EALDH1A1PPARG
SCHEMBL9348996 0.64 PTGS1 (0.76) PTGS2PTGS1ALOX5
SCHEMBL9122974 0.60 PTGS1 (0.40) PTGS2PTGS1
SCHEMBL9120689 0.60 PTGS1 (0.35) PTGS2PTGS1
SCHEMBL9738006 0.60 PTGS1 (0.58) PTGS2PTGS1ALOX5GAA
SCHEMBL3618030 0.59 PTGS1 (0.40) PTGS2PTGS1ALDH1A1SMN1; SMN2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356898-A Antiinflammatory agents, antiallergens, antiulcer agents WARNER-LAMBERT COMPANY (US) 1994-10-18 US claimed
US-5432181-A Substituted heteroaryl analogs of 4,6-di-tertiary-butyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1995-07-11 US disclosed
US-5356898-A Antiinflammatory agents, antiallergens, antiulcer agents WARNER-LAMBERT COMPANY (US) 1994-10-18 US disclosed
WO-1992013844-A1 SUBSTITUTED 4,6-DI-TERTIARY-BUTYL-5-HYDROXY-PYRIMIDINES WARNER-LAMBERT COMPANY (US) 1992-08-20 WO disclosed