SCHEMBL9119840

SCHEMBL9119840

COc1ccc(C(=O)CCCCBr)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 3/20 0.65
WNT3A P56704 3/20 0.65
MAPT P10636 3/20 0.56
TSHR P16473 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
ALDH1A1 P00352 3/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA7 P43166 1/20 0.54
TPMT P51580 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
ACHE P22303 1/20 0.53
PAX8 Q06710 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27200216 0.98 CTNNB1 (0.63) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL5355533 0.98 CTNNB1 (0.63) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL31556192 0.93 CTNNB1 (0.73) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL31556194 0.92 CTNNB1 (0.71) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL14483927 0.90 CTNNB1 (0.69) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL9375696 0.87 CTNNB1 (0.65) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL9557967 0.86 HPGD (0.51) CTNNB1WNT3ACYP1A2CYP2C19ALDH1A1
SCHEMBL10455919 0.86 CTNNB1 (0.83) CTNNB1WNT3AMAPTTSHRCYP1A2
SCHEMBL9588048 0.86 THRA (0.66) CTNNB1WNT3APDE4BPDE4APDE4C
SCHEMBL9117986 0.86 CTNNB1 (0.63) CTNNB1WNT3AMAPTTSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548664-B1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives HOFFMANN LA ROCHE (CH) 1995-05-31 EP disclosed
US-5318967-A Cognition activators for alzheimer's disease, learning enhancement HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
US-5318966-A Administering the enzyme inhibitor for treating alzheimer's disease, learning enhancement, brain disorders HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
EP-0548664-A1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed