SCHEMBL9119923

SCHEMBL9119923

CC1=C(C(=O)O)C(c2cccc(F)c2)C(C(=O)O)=C(C)N1C

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.50
NPSR1 Q6W5P4 3/20 0.50
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.48
KMT2A Q03164 1/20 0.47
CACNA1B Q00975 1/20 0.46
LMNA P02545 2/20 0.45
NOTUM Q6P988 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
HTR7 P34969 1/20 0.40
PDE5A O76074 1/20 0.39
RIPK1 Q13546 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9121128 0.84 TSHR (0.71) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL16178460 0.84 TSHR (0.43) TSHRNPSR1KDM4EGAACACNA1B
SCHEMBL11753470 0.84 CACNA1B (0.55) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL16178523 0.82 KDM4E (0.66) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL16178473 0.81 MET (0.49) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL16178557 0.81 TSHR (0.50) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL8699921 0.80 CACNA1B (0.65) KMT2ACACNA1B
SCHEMBL10656803 0.77 CACNA1F (0.53) TSHRNPSR1KMT2ACACNA1BLMNA
SCHEMBL11750748 0.77 KDM4E (0.53) TSHRNPSR1KDM4EGAAKMT2A
SCHEMBL9363842 0.75 KMT2A (0.47) TSHRNPSR1KMT2ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5432185-A Treating patients exhibiting acute or chronic ischaemic disorders associated with disorders of microcirculation, without lowering or increasing blood pressure BAYER AKTIENGESELLSCHAFT (DE) 1995-07-11 US disclosed
US-5234935-A Preventing myocardial infarct BAYER AKTIENGESELLSCHAFT (DE) 1993-08-10 US disclosed