SCHEMBL9119962

SCHEMBL9119962

Oc1ccc(Cl)cc1-n1c(=S)[nH]c2cc(C(F)(F)F)ccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.60
CYP3A4 P08684 4/20 0.60
CYP2C19 P33261 4/20 0.60
HSP90AA1 P07900 2/20 0.60
CYP1A2 P05177 2/20 0.60
MAPT P10636 2/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
TSHR P16473 1/20 0.60
NFKB1 P19838 1/20 0.60
BLM P54132 1/20 0.60
PMP22 Q01453 1/20 0.60
KCNMA1 Q12791 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
ALDH1A1 P00352 4/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
KCNH2 Q12809 1/20 0.46
CYP2D6 P10635 2/20 0.40
CHRNA7 P36544 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8654682 0.91 HSP90AA1 (0.71) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL29948904 0.85 HSP90AA1 (0.83) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL3102522 0.85 HSP90AA1 (0.83) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL29748943 0.85 HSP90AA1 (0.83) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL9119844 0.84 KMT2A (0.57) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL9119253 0.82 ALDH1A1 (0.48) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL9119790 0.81 KMT2A (0.54) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL5632986 0.81 HSP90AA1 (0.83) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL2820871 0.76 HSP90AA1 (1.00) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2
SCHEMBL29630342 0.76 HSP90AA1 (1.00) CYP2C9CYP3A4CYP2C19HSP90AA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477819-B1 Benzimidazole derivatives, their preparation and use NEUROSEARCH AS (DK) 1995-03-15 EP disclosed
US-5200422-A Benzimidazole derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-04-06 US disclosed
EP-0477819-A2 Benzimidazole derivatives, their preparation and use NEUROSEARCH A/S (DK) 1992-04-01 EP disclosed