SCHEMBL9124265

SCHEMBL9124265

Nc1ncccc1OCc1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.60
MAPK14 Q16539 1/20 0.60
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
HTT P42858 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
MAPT P10636 1/20 0.51
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MET P08581 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
DCPS Q96C86 3/20 0.35
DHFR P00374 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9123661 0.85 LTA4H (0.55) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL488298 0.85 LTA4H (0.58) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL3019351 0.84 LTA4H (0.54) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL9127353 0.82 MAPK14 (0.55) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL488397 0.80 LTA4H (0.53) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL6079578 0.79 LTA4H (0.75) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL488813 0.79 RAB9A (0.55) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL488951 0.78 NPC1 (0.61) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL9747086 0.78 LTA4H (0.58) LTA4HMAPK14NPC1RAB9AHTT
SCHEMBL6079764 0.78 LTA4H (0.54) LTA4HMAPK14NPC1RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed