SCHEMBL9126133

SCHEMBL9126133

COc1ccc(COc2cccnc2N)c(F)c1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.63
RAB9A P51151 3/20 0.63
CSF1R P07333 1/20 0.48
LTA4H P09960 1/20 0.48
MAPK14 Q16539 1/20 0.48
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
GRM2 Q14416 2/20 0.43
SYK P43405 3/20 0.42
PARP10 Q53GL7 2/20 0.42
PARP14 Q460N5 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
P2RX7 Q99572 1/20 0.41
CHRNA7 P36544 1/20 0.40
ABCB1 P08183 1/20 0.40
USP7 Q93009 1/20 0.40
MTNR1B P49286 1/20 0.40
PARP15 Q460N3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080485 0.85 MAPK14 (0.54) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL6079375 0.79 LTA4H (0.61) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL9125665 0.77 NPC1 (1.00) NPC1RAB9ACSF1RLTA4HMAPK14
SCHEMBL9115564 0.77 NPC1 (0.72) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL6080009 0.76 NPC1 (0.61) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL488182 0.74 RAB9A (0.58) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL13529594 0.74 CSF1R (0.44) NPC1RAB9ACSF1RCHRNA7USP7
SCHEMBL6079764 0.73 LTA4H (0.54) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL9127353 0.72 MAPK14 (0.55) NPC1RAB9ALTA4HMAPK14MAPT
SCHEMBL9126648 0.71 LTA4H (0.51) NPC1RAB9ALTA4HMAPK14MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed