SCHEMBL9130285

SCHEMBL9130285

COCCC1=CCN(C)CC1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
QDPR P09417 3/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9129342 0.82 QDPR (0.43) QDPRALDH1A1KMT2A
SCHEMBL9644027 0.79 QDPR (0.39) QDPR
SCHEMBL13783321 0.77 QDPR (0.42) QDPR
SCHEMBL13599361 0.76 QDPR (0.37) QDPRCHRM2CHRM4CHRM5CHRM1
SCHEMBL4426898 0.75 HRH3 (0.38) QDPRALDH1A1KMT2ACHRM2CHRM4
SCHEMBL6947872 0.74 QDPR (0.36) QDPR
SCHEMBL3424079 0.74 QDPR (0.40) QDPR
SCHEMBL10752307 0.74 QDPR (0.36) QDPRCHRM2CHRM4CHRM5CHRM1
SCHEMBL9127424 0.74 QDPR (0.36) QDPR
SCHEMBL7607024 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325263-B1 TETRAHYDROPYRIDINE DERIVATIVES BOEHRINGER INGELHEIM KG (DE) 1992-09-23 EP claimed
EP-0325263-A1 Tetrahydropyridine derivatives BOEHRINGER INGELHEIM KG (DE) 1989-07-26 EP claimed
US-5422353-A Alzheimer*s disease, glaucoma treatment BOEHRINGER INGELHEIM KG (DE) 1995-06-06 US disclosed
EP-0325263-B1 TETRAHYDROPYRIDINE DERIVATIVES BOEHRINGER INGELHEIM KG (DE) 1992-09-23 EP disclosed
EP-0325263-A1 Tetrahydropyridine derivatives BOEHRINGER INGELHEIM KG (DE) 1989-07-26 EP disclosed