SCHEMBL9130664

SCHEMBL9130664

C=CCOc1ccc(C(=O)Cl)cc1OCC=C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
TSHR P16473 3/20 0.51
GAA P10253 1/20 0.51
PDE4B Q07343 1/20 0.48
LIG1 P18858 1/20 0.42
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KMT2A Q03164 2/20 0.39
CYP2D6 P10635 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FLT3 P36888 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11226244 0.87 KDM4E (0.55) KDM4ETSHRGAAPDE4BLIG1
SCHEMBL15312851 0.85 KDM4E (0.60) KDM4ETSHRGAAPDE4BALDH1A1
SCHEMBL22229873 0.83 KDM4E (0.62) KDM4ETSHRGAAPDE4BLIG1
SCHEMBL13690626 0.82 KDM4E (0.57) KDM4ETSHRGAAPDE4BLIG1
SCHEMBL19815469 0.81 KDM4E (0.46) KDM4ETSHRGAAPDE4BLIG1
SCHEMBL4331415 0.80 KDM4E (0.55) KDM4ETSHRGAAPDE4BLIG1
SCHEMBL4363165 0.77 KMT2A (0.43) TSHRALDH1A1LMNAKMT2AMEN1
SCHEMBL711175 0.77 NPC1 (0.54) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL184107 0.77 TSHR (0.60) KDM4ETSHRALDH1A1HPGDLMNA
SCHEMBL8484361 0.76 KDM4E (0.66) KDM4ETSHRGAAPDE4BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2290839-A None JP disclosed
US-5447925-A Carbapenems with side-chain S; use to treat infections IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-09-05 US disclosed
EP-0580632-A1 ANTIBIOTIC CARBAPENEM DERIVATIVES ZENECA LIMITED (GB) 1994-02-02 EP disclosed
WO-1992017480-A1 ANTIBIOTIC CARBAPENEM DERIVATIVES ZENECA LTD. (GB) 1992-10-15 WO disclosed
JP-H02290839-A ESTER DERIVATIVE MITSUBISHI KASEI CORP 1990-11-30 JP disclosed