SCHEMBL913262

SCHEMBL913262

c1cnc(C2CNCCO2)nc1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrogen Sulfide SCHEMBL28070942 0.98 DRD2 (0.45) DRD2DRD3HTR1A
Sulfur Dioxide SCHEMBL28071143 0.93 DRD2 (0.42) DRD2DRD3HTR1A
Guanidine SCHEMBL28415570 0.90 DRD2 (0.43) DRD2DRD3HTR1A
SCHEMBL27547345 0.83 DRD2 (0.41) DRD2DRD3
SCHEMBL8143198 0.81 DRD2 (0.41) DRD2DRD3
SCHEMBL28648650 0.80 DRD2 (0.50) DRD2DRD3
SCHEMBL17224079 0.80
SCHEMBL17224077 0.80
SCHEMBL28289256 0.80
SCHEMBL28679348 0.79 DRD2 (0.43) DRD2DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 106 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102952086-B Preparation method of 2-morpholinyl-substituted pyrimidine compounds TIANJIN SCIPHARMACN LTD 2013-08-28 CN claimed
CN-101553233-A Kinase inhibitors useful for the treatment of myleoproliferative diseases and other proliferative diseases DECIPHERA PHARMACEUTICALS LLC (US) 2009-10-07 CN claimed
CN-101553232-A Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS LLC (US) 2009-10-07 CN claimed
CN-101516379-A Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS LLC (US) 2009-08-26 CN claimed
WO-2025133334-A1 NOVEL VDAC1 INHIBITORS ABARCEO PHARMA AB (SE) 2025-06-26 WO disclosed
CN-111303048-B Pyrimidine guanidine compound, and preparation method and application thereof 沈阳农业大学 2023-05-26 CN disclosed
CN-110461842-A FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB BIOPHARMA SPRL 2019-11-15 CN disclosed
CN-107108672-B Condensed five rings imdazole derivatives UCB生物制药私人有限公司 2019-11-08 CN disclosed
CN-105814043-B Triazolopyridine derivatives as TNF active regulator UCB生物制药私人有限公司 2019-05-17 CN disclosed
CN-105814049-B Fused tricyclic imdazole derivatives as TNF active regulator UCB生物制药私人有限公司 2019-03-12 CN disclosed
CN-109219608-A FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-15 CN disclosed
CN-109219609-A FUSED HEXACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-15 CN disclosed
WO-2005000404-A2 HETEROCYCLIC COMPOUNDS FOR PREVENTING AND TREATING DISORDERS ASSOCIATED WITH EXCESSIVE BONE LOSS SYNTA PHARMACEUTICALS, CORP. (US) 2005-01-06 WO disclosed
US-20040053937-A1 Pyrimidine compounds SYNTA PHARMACEUTICALS CORP. 2004-03-18 US disclosed
US-20040048873-A1 Pyrimidine compounds SYNTA PHARMACEUTICALS CORP., A DELAWARE CORPORATIO 2004-03-11 US disclosed
US-6693097-B2 Pyrimidine compounds SYNTA PHARMACEUTICALS CORP. 2004-02-17 US disclosed
US-20040024206-A1 Pyrimidine compounds MADRIGAL PHARMACEUTICALS, INC. 2004-02-05 US disclosed
US-6660733-B2 Induce immunology response SYNTA PHARMACEUTICALS CORP. 2003-12-09 US disclosed
US-20030139403-A1 Pyrimidine compounds SHIONOGI BIORESEARCH CORP. 2003-07-24 US disclosed
US-20030114446-A1 Pyrimidine compounds SYNTA PHARMACEUTICALS CORP. 2003-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053937-A1 Pyrimidine compounds CCNO, CNR1, CBR1 DRD2 567/4885DRD3 828/4885HTR1A 645/4885
US-20030139403-A1 Pyrimidine compounds CBR1, CBR3, CCNO DRD2 75/4885DRD3 124/4885HTR1A 1705/4885
US-20030114446-A1 Pyrimidine compounds CCNO, CNR1, CBR1 DRD2 570/4885DRD3 778/4885HTR1A 686/4885
US-20040024206-A1 Pyrimidine compounds CBR1, CCR4, CNR1 DRD2 524/4885DRD3 617/4885HTR1A 2249/4885
US-20040048873-A1 Pyrimidine compounds CBR1, CBR3, CCNO DRD2 68/4885DRD3 101/4885HTR1A 1889/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.