SCHEMBL9138797

SCHEMBL9138797

NCC[C@@H]1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
ATM Q13315 1/20 0.41
CCR5 P51681 2/20 0.40
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.38
IDO1 P14902 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7805572 0.94 TDP1 (0.42) TDP1ATMCCR5RAB9ANPC1
SCHEMBL8781804 0.91 TDP1 (0.42) TDP1ATMCCR5RAB9ANPC1
SCHEMBL7805543 0.91 TDP1 (0.43) TDP1ATMCCR5RAB9ANPC1
SCHEMBL9137735 0.90 CCR5 (0.43) TDP1ATMCCR5RAB9AALDH1A1
SCHEMBL8781845 0.90 CCR5 (0.40) TDP1ATMCCR5RAB9ANPC1
SCHEMBL7858569 0.88 TDP1 (0.41) TDP1ATMCCR5RAB9ANPC1
SCHEMBL9363174 0.87 CCR5 (0.42) TDP1ATMCCR5
SCHEMBL8782026 0.87 CCR5 (0.39) TDP1ATMCCR5RAB9ANPC1
SCHEMBL7811544 0.87 CCR5 (0.41) TDP1ATMCCR5RAB9ANPC1
SCHEMBL9519179 0.86 TDP1 (0.42) TDP1ATMCCR5RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449672-A Bactericides BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-09-12 US disclosed
EP-0544307-A1 Alkylaminoakylpyrrolidinylthiocarbapenem derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-02 EP disclosed