SCHEMBL9147485

SCHEMBL9147485

COS(=O)(=O)c1ccc2cc(S(=O)(=O)OC)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.46
LMNA P02545 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PKM P14618 1/20 0.43
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
TSHR P16473 3/20 0.41
KDM4E B2RXH2 2/20 0.41
PLAU P00749 1/20 0.41
CASP1 P29466 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29732529 0.92 L3MBTL1 (0.57) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL3633735 0.92 L3MBTL1 (0.57) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL16467640 0.88 CYP1A2 (0.42) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL15352702 0.88 CYP2A6 (0.42) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL16467682 0.88 CYP2A6 (0.42) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL6530359 0.88 HTR6 (0.42) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL28740645 0.87 L3MBTL1 (0.57) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL16467719 0.82 CYP2A6 (0.41) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL16467726 0.82 CYP1A2 (0.41) L3MBTL1LMNATDP1HTTSMN1; SMN2
SCHEMBL15352636 0.82 CYP2A6 (0.41) L3MBTL1LMNATDP1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2843473-B1 Toner CANON KK (JP) 2016-11-02 EP disclosed
US-9229345-B2 Toner CANON KABUSHIKI KAISHA (JP) 2016-01-05 US disclosed
CN-104423185-A Toner CANON KK 2015-03-18 CN disclosed
EP-2843473-A1 Toner Canon Kabushiki Kaisha (JP) 2015-03-04 EP disclosed
US-20150056549-A1 TONER CANON KABUSHIKI KAISHA (JP) 2015-02-26 US disclosed
EP-0625971-A4 UV LIGHT STABILIZING, ANTIOXIDANT AND COLORANT COMPOUNDS. 1995-01-04 EP disclosed
EP-0625971-A1 UV LIGHT STABILIZING, ANTIOXIDANT AND COLORANT COMPOUNDS HOECHST CELANESE CORPORATION (US) 1994-11-30 EP disclosed
WO-1993015063-A1 UV LIGHT STABILIZING, ANTIOXIDANT AND COLORANT COMPOUNDS HOECHST CELANESE CORPORATION (US) 1993-08-05 WO disclosed
US-4434104-A REACTING NAPHTHALENEDISULFONATE CHLORIDE AND EXCESS ALCOHOL, TREATING WITH ALKALI METAL ALCOHOLATE AND WASHING NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1984-02-28 US disclosed