SCHEMBL9148643

SCHEMBL9148643

CCCCc1nn(Cc2ccccc2)c(=O)n1Cc1ccc(NS(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.55
AGTR1 P30556 3/20 0.53
AGTR2 P50052 3/20 0.53
NR3C1 P04150 1/20 0.49
PPARG P37231 1/20 0.49
PPARD Q03181 1/20 0.49
ESR2 Q92731 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3627824 0.76 AGTR2 (0.56) AGTR2
SCHEMBL3631709 0.76 AGTR1 (0.58) AGTR1AGTR2
SCHEMBL9031922 0.75 AGTR1 (0.61) AGTR1AGTR2
SCHEMBL9141157 0.72 AGTR1 (0.67) AGTR1
SCHEMBL647 0.71
SCHEMBL1258786 0.70 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL1258665 0.70 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL1257529 0.70 AGTR2 (0.47) AGTR2
SCHEMBL1257795 0.70 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL9166785 0.70 AGTR1 (1.00) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5411980-A Substituted triazolinones, triazolinethiones, and triazolinimines as angiotensin II antagonists MERCK & CO., INC. (US) 1995-05-02 US disclosed