SCHEMBL9150359

SCHEMBL9150359

CCCCCc1ccc(-c2ccc(C#N)c(F)c2)nc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.54
NPC1 O15118 6/20 0.54
SMN1; SMN2 Q16637 5/20 0.54
MAPT P10636 2/20 0.54
STAT3 P40763 1/20 0.54
ATM Q13315 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.53
NFKB1 P19838 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
MAPK1 P28482 1/20 0.53
CASP3 P42574 2/20 0.53
SENP8 Q96LD8 2/20 0.53
SENP7 Q9BQF6 2/20 0.53
SENP6 Q9GZR1 2/20 0.53
TP53 P04637 1/20 0.52
PKM P14618 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CYP11B1 P15538 8/20 0.47
CYP11B2 P19099 8/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9151076 0.99 RAB9A (0.56) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL9152695 0.99 RAB9A (0.56) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL7910603 0.99 RAB9A (0.56) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL9151651 0.99 RAB9A (0.56) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL9151358 0.99 RAB9A (0.56) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL9151591 0.96 RAB9A (0.58) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL8377173 0.92 RAB9A (0.54) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL9151552 0.91 NPC1 (0.62) RAB9ANPC1SMN1; SMN2L3MBTL1NFKB1
SCHEMBL10716920 0.88 RAB9A (0.47) RAB9ANPC1SMN1; SMN2MAPTSTAT3
SCHEMBL10359182 0.87 RAB9A (0.57) RAB9ANPC1SMN1; SMN2MAPTSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252961-B1 HETEROCYCLIC COMPOUNDS AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GMBH (DE) 1995-02-08 EP claimed
EP-0252961-B1 HETEROCYCLIC COMPOUNDS AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GMBH (DE) 1995-02-08 EP disclosed
US-4913837-A Heterocyclic compounds MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-04-03 US disclosed