SCHEMBL9150800

SCHEMBL9150800

CCCc1cc2c(cc1CCO)OCO2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.53
ALDH1A1 P00352 4/20 0.53
TSHR P16473 1/20 0.53
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP2D6 P10635 4/20 0.44
CYP1A2 P05177 3/20 0.44
CYP2C19 P33261 3/20 0.44
CYP2C9 P11712 2/20 0.44
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 1/20 0.43
HPGD P15428 1/20 0.38
KDM4E B2RXH2 1/20 0.38
SCN1A P35498 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN3A Q9NY46 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL352250 0.88 CYP3A4 (0.53) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL9150522 0.88 CYP3A4 (0.41) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL9678088 0.83 CYP3A4 (0.56) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL30927115 0.83 CYP3A4 (0.56) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL1276072 0.80 CYP3A4 (0.49) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL9148130 0.80 CYP3A4 (0.53) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL9150579 0.80 ALDH1A1 (0.38) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL128215 0.78 CYP3A4 (0.73) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL30927087 0.78 CYP3A4 (0.73) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL9148810 0.78 MEN1 (0.48) CYP3A4ALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475024-A Useful in treating liver disease EISAI CO., LTD. (JP) 1995-12-12 US disclosed
US-5292901-A Benzodioxole derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
EP-0281098-B1 BENZODIOXOLE DERIVATIVES, COMPOSITIONS COMPRISING THE SAME, AND THE USE OF THE SAME FOR THE MANUFACTURE OF MEDICAMENTS Eisai Co., Ltd. (JP) 1992-11-25 EP disclosed
US-5110956-A Liver disorders EISAI CO., LTD. (JP) 1992-05-05 US disclosed
EP-0281098-A1 Benzodioxole derivatives, compositions comprising the same, and the use of the same for the manufacture of medicaments Eisai Co., Ltd. (JP) 1988-09-07 EP disclosed