SCHEMBL9150944

SCHEMBL9150944

N#Cc1ccc2c(c1)C(O)CCO2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 2/20 0.47
DRD2 P14416 7/20 0.41
DRD3 P35462 7/20 0.41
HCRTR2 O43614 1/20 0.39
CYP2D6 P10635 2/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ABCB1 P08183 2/20 0.38
ABCC9 O60706 3/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.38
CHRNA1 P02708 1/20 0.37
CHRNG P07510 1/20 0.37
CHRNB1 P11230 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9585693 0.91 DRD2 (0.40) MAP3K14DRD2DRD3HCRTR2CYP2D6
SCHEMBL4140398 0.87 MAP3K14 (0.59) MAP3K14DRD2DRD3CHRNA1CHRNG
SCHEMBL4133966 0.87 MAP3K14 (0.59) MAP3K14DRD2DRD3CHRNA1CHRNG
SCHEMBL29243618 0.82 DRD2 (0.42) DRD2DRD3HCRTR2ABCB1CHRNA1
SCHEMBL1266045 0.82 DRD2 (0.42) DRD2DRD3HCRTR2ABCB1CHRNA1
SCHEMBL9585392 0.82 DRD2 (0.38) DRD2DRD3HCRTR2CYP2D6KDM4E
SCHEMBL9585396 0.82 DRD2 (0.38) DRD2DRD3HCRTR2CYP2D6KDM4E
SCHEMBL9585384 0.82 DRD2 (0.38) DRD2DRD3HCRTR2CYP2D6KDM4E
SCHEMBL24075797 0.81 DRD2 (0.44) DRD2DRD3HCRTR2ABCB1CHRNA1
SCHEMBL24090487 0.81 DRD2 (0.44) DRD2DRD3HCRTR2ABCB1CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447943-A Smooth muscle relaxants or bronchodilators SYNTEX (U.S.A.) INC. (US) 1995-09-05 US disclosed
US-5250547-A Potassium channel activators; 5-lipoxygenase inhibitors; muscle relaxants; bronchodilators SYNTEX (U.S.A.) INC. (US) 1993-10-05 US disclosed
EP-0529654-A1 Benzopyran derivatives as potassium channel activators and 5-lipoxygenase inhibitors SYNTEX (U.S.A.) INC. (US) 1993-03-03 EP disclosed