SCHEMBL9154751

SCHEMBL9154751

C=CCN1CCC[C@H]1CN

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.38
DRD3 P35462 7/20 0.36
DRD4 P21917 6/20 0.36
HTR1A P08908 3/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD1 P21728 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
KCNH2 Q12809 1/20 0.35
CA9 Q16790 1/20 0.35
CA13 Q8N1Q1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5804458 1.00 DRD2 (0.38) DRD2DRD3DRD4HTR1ACA12
SCHEMBL8649163 0.94 DRD2 (0.34) DRD2DRD3DRD4HTR1ACA12
Isothiocyanate SCHEMBL11011138 0.90 DRD2 (0.34) DRD2DRD3DRD4HTR1ACA12
SCHEMBL7372904 0.85 DRD2 (0.36) DRD2DRD3DRD4HTR1ACA12
SCHEMBL8799867 0.82 CHRNB2 (0.37) DRD2DRD3DRD4HTR1ACA12
SCHEMBL8436147 0.80 POLB (0.42) DRD2DRD3DRD4HTR1ACA12
SCHEMBL11445454 0.80 DRD2 (0.36) DRD2DRD3DRD4HTR1ACA12
SCHEMBL11300057 0.80 POLB (0.42) DRD2DRD3DRD4HTR1ACA12
SCHEMBL11251940 0.80 DRD2 (0.36) DRD2DRD3DRD4HTR1ACA12
SCHEMBL9036814 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1298702-C Process for preparing (s)-1-allyl-2-amidomethyl tetrahydropyrrole JIANGSU PROV ATOM MEDICINE INS (CN) 2007-02-07 CN disclosed
CN-1298702-C Process for preparing (s)-1-allyl-2-amidomethyl tetrahydropyrrole JIANGSU PROV ATOM MEDICINE INS (CN) 2007-02-07 CN disclosed
CN-1683335-A Process for preparing (S)-1-allyl-2-amidomethyl tetrahydropyrrole JIANGSU PROV ATOM MEDICINE INS (CN) 2005-10-19 CN disclosed
CN-1683335-A Process for preparing (S)-1-allyl-2-amidomethyl tetrahydropyrrole JIANGSU PROV ATOM MEDICINE INS (CN) 2005-10-19 CN disclosed
US-5468876-A Intermediates for the stereoconservative synthesis of 1-substituted (S)-and (R)-2-aminomethylpyrrolidines AKTIEBOLAGET ASTRA (SE) 1995-11-21 US disclosed
US-5300660-A Efficient stereoconservative synthesis of 1-substituted (S)- and (R)-2-aminomethylpyrrolidines and intermediates thereto ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1994-04-05 US disclosed
EP-0253785-B1 EFFICIENT STEREOCONSERVATIVE SYNTHESES OF 1-SUBSTITUTED (S)- AND (R)-2-AMINOMETHYLPYRROLIDINES AND INTERMEDIATES THEREIN ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1992-11-11 EP disclosed
EP-0270596-A1 A STEREOCONSERVATIVE SYNTHESIS OF 1-SUBSTITUTED (S)- AND (R)-2-AMINOMETHYLPYRROLIDINES AND INTERMEDIATES THERETO ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1988-06-15 EP disclosed
WO-1987007271-A1 A STEREOCONSERVATIVE SYNTHESIS OF 1-SUBSTITUTED (S)- AND (R)-2-AMINOMETHYLPYRROLIDINES AND INTERMEDIATES THERETO Astra Läkemedel Aktiebolag (SE) 1987-12-03 WO disclosed