SCHEMBL9156972

SCHEMBL9156972

COc1ccc2ncc(O)cc2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
F2 P00734 1/20 0.62
GLA P06280 1/20 0.62
HPGD P15428 1/20 0.62
PDGFRB P09619 6/20 0.58
PDGFRA P16234 6/20 0.58
EGFR P00533 3/20 0.57
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
MAP4K4 O95819 1/20 0.50
CDK8 P49336 1/20 0.50
CLK2 P49760 1/20 0.50
CDK7 P50613 1/20 0.50
CDK9 P50750 1/20 0.50
CDK5 Q00535 1/20 0.50
ACVR1 Q04771 1/20 0.50
ROCK1 Q13464 1/20 0.50
DYRK1A Q13627 1/20 0.50
LRRK2 Q5S007 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL620457 0.86 ALDH1A1 (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL7028923 0.85 ALDH1A1 (0.70) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL18250877 0.83 MAP4K4 (0.47) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL434861 0.80 PDGFRB (0.59) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL444746 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL27918947 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL621672 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL27930034 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL1928147 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB
SCHEMBL20033882 0.79 PDGFRB (0.58) ALDH1A1F2GLAHPGDPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5442065-A Antitumor agents BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1995-08-15 US disclosed
US-5442065-A Antitumor agents BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1995-08-15 US disclosed